Table 3
Interaction between CYPs and olanzapine
Enzyme
Involved in metabolism of olanzapine
Inhibited by olanzapine; in vitro data only
In vitro
In vivo
Case reports
Case series
CYP1A2
+
+
+
−
CYP2C9
−
CYP2D6
+
+ (NC)
−
CYP3A4
−
−