Table 2
Interaction between CYPs and risperidone
Enzyme
Involved in metabolism of risperidone
Inhibited by risperidone; in vitro data only
In vitro
In vivo
Case reports
Case series
CYP1A1
−
CYP1A2
−
−
CYP2C9
−
−
CYP2C19
−
−
CYP2D6
+
+
+
+ (NC)
CYP3A4
+/−
+
+
−