Table 2

Interaction between CYPs and risperidone

EnzymeInvolved in metabolism of risperidoneInhibited by risperidone; in vitro data only
In vitroIn vivo
Case reportsCase series
CYP1A1
CYP1A2
CYP2C9
CYP2C19
CYP2D6++++ (NC)
CYP3A4+/−++