Predicting drug interactions and pharmacokinetic variability with in vitro methods: the olanzapine experience

Drug Metab Rev. 1999 Feb;31(1):15-28. doi: 10.1081/dmr-100101905.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Antipsychotic Agents / metabolism
  • Antipsychotic Agents / pharmacokinetics*
  • Benzodiazepines
  • Cytochrome P-450 Enzyme System / isolation & purification
  • Cytochrome P-450 Enzyme System / metabolism*
  • Drug Interactions
  • Humans
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / enzymology
  • Microsomes, Liver / metabolism
  • Olanzapine
  • Pirenzepine / analogs & derivatives*
  • Pirenzepine / metabolism
  • Pirenzepine / pharmacokinetics

Substances

  • Antipsychotic Agents
  • Benzodiazepines
  • Pirenzepine
  • Cytochrome P-450 Enzyme System
  • Olanzapine